17/09/2019
Our team in collaboration with AstraZeneca developed an integrative systems pharmacology model of lipoprotein homeostasis which sets the stage for the quantitative benchmarking of two anti-PCSK9 pharmacological modality classes, monoclonal antibodies, and small interfering RNA, by describing in minimalistic yet mechanistic terms complex interactions between multiple plasma lipoprotein and lipid biomarkers, and by establishing a quantitative link between plasma PCSK9 and low-density lipoprotein cholesterol reduction for five different anti-PCSK9 compounds.